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This website is a work-in-progress and is actively being developed. As such the user experience may have room for improvement, or content may be incomplete.
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Supplemental Information
Screen Description
Export
Kinase HTS
Barcodes
Kinase HTS
Screen Structure
Kinase HTS
Well Count | 96 |
---|---|
Number of distinct ingredients | 64 |
Internal diversity (score mean dist) | 0.936 |
Screen Composition
ingredient type | Kinase HTS |
---|---|
Buffer | 111 |
Cryoprotectant | 3 |
Organic (non-volatile) | 20 |
Organic (volatile) | 6 |
Polymer | 77 |
Salt | 101 |
Well Contents
Buffers are shown in italics.
More information about buffers.
Primary factors are shown in bold.
More information about primary factors.
Well | Ingredient, Concentration, Units, pH | pH | Recipe 1000μl |
---|---|---|---|
A1 |
| pH 5.6 | 100 μl of tri-Sodium citrate pH 5.6 (1 M) 333 μl of Ammonium sulfate (3 M) 100 μl of Magnesium acetate (2 M) 100 μl of Dithiothreitol (0.1 M) 366 μl of water (100 v/v) |
A2 |
| pH 5.6 | 100 μl of tri-Sodium citrate pH 5.6 (1 M) 433 μl of Ammonium sulfate (3 M) 466 μl of water (100 v/v) |
A3 |
| pH 8.5 | 433 μl of Ammonium sulfate (3 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 466 μl of water (100 v/v) |
A4 |
| pH 6.5 | 25 μl of Cobalt (II) chloride (1 M) 100 μl of MES pH 6.5 (1 M) 600 μl of Ammonium sulfate (3 M) 275 μl of water (100 v/v) |
A5 |
| pH 3.1 | 100 μl of tri-Sodium citrate pH 3.1 (1 M) 200 μl of Sodium chloride (1 M) 666 μl of Ammonium sulfate (3 M) 33 μl of water (100 v/v) |
A6 |
| pH 4.6 | 20 μl of Magnesium chloride (2.5 M) 100 μl of Sodium acetate pH 4.6 (1 M) 666 μl of Ammonium sulfate (3 M) 213 μl of water (100 v/v) |
A7 |
| pH 4.6 | 100 μl of Sodium acetate pH 4.6 (1 M) 666 μl of Ammonium sulfate (3 M) 233 μl of water (100 v/v) |
A8 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 20 μl of Polyethylene glycol monomethyl ether 550 (100 v/v) 666 μl of Ammonium sulfate (3 M) 213 μl of water (100 v/v) |
A9 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 666 μl of Ammonium sulfate (3 M) 233 μl of water (100 v/v) |
A10 |
| pH 8.5 | 2 μl of Magnesium chloride (2.5 M) 666 μl of Ammonium sulfate (3 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 230 μl of water (100 v/v) |
A11 |
| pH 8.5 | 2 μl of Nickel sulfate (4 M) 500 μl of Lithium sulfate (3 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 397 μl of water (100 v/v) |
A12 |
| pH 4.2 | 200 μl of Lithium chloride (5 M) 100 μl of tri-Sodium citrate pH 4.2 (1 M) 700 μl of water (100 v/v) |
B1 |
| pH 4.6 | 400 μl of Sodium chloride (5 M) 100 μl of Sodium acetate pH 4.6 (1 M) 500 μl of water (100 v/v) |
B2 |
| pH 6.5 | 50 μl of Potassium di-hydrogen phosphate (2 M) 400 μl of Sodium chloride (5 M) 100 μl of MES pH 6.5 (1 M) 20 μl of di-Sodium hydrogen phosphate (5 M) 430 μl of water (100 v/v) |
B3 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 660 μl of Sodium chloride (5 M) 10 μl of Glycerol (100 v/v) 230 μl of water (100 v/v) |
B4 |
| pH 6.5 | 600 μl of Sodium acetate (2 M) 62 μl of Calcium chloride (1 M) 100 μl of MES pH 6.5 (1 M) 237 μl of water (100 v/v) |
B5 |
| pH 9.5 | 528 μl of Sodium formate (7 M) 40 μl of Polyethylene glycol 3,000 (50 w/v) 100 μl of BICINE pH 9.5 (1 M) 331 μl of water (100 v/v) |
B6 |
| pH 6 | 166 μl of di-Sodium malonate pH 6 (3 M) 50 μl of PIPES pH 6 (1 M) 16 μl of Glycerol (100 v/v) 100 μl of Dithiothreitol (0.1 M) 667 μl of water (100 v/v) |
B7 |
| pH 10 | 100 μl of CAPS pH 10 (1 M) 250 μl of Potassium di-hydrogen phosphate (2 M) 66 μl of Lithium sulfate (3 M) 100 μl of di-Sodium hydrogen phosphate (5 M) 483 μl of water (100 v/v) |
B8 |
| pH 8.5 | 600 μl of di-Sodium tartrate (2 M) 50 μl of Dithiothreitol (0.1 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 250 μl of water (100 v/v) |
B9 |
| pH 6.5 | 500 μl of Potassium Sodium tartrate (2 M) 100 μl of MES pH 6.5 (1 M) 400 μl of water (100 v/v) |
B10 |
| pH 6.5 | 50 μl of Cesium chloride (1 M) 600 μl of Jeffamine® M-600 (50 v/v) 100 μl of MES pH 6.5 (1 M) 250 μl of water (100 v/v) |
B11 |
| pH 6.5 | 400 μl of 2-methyl-2,4-pentanediol BCC (100 v/v) 100 μl of MES pH 6.5 (1 M) 500 μl of water (100 v/v) |
B12 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 500 μl of 2-methyl-2,4-pentanediol BCC (100 v/v) 400 μl of water (100 v/v) |
C1 |
| pH 8.5 | 142 μl of Ethylenediaminetetraacetic acid disodium salt (7 mM) 60 μl of Sodium chloride (5 M) 100 μl of Polyethylene glycol 400 (100 v/v) 10 μl of Dithiothreitol (0.1 M) 50 μl of tris chloride BCC pH 8.5 (1 M) 637 μl of water (100 v/v) |
C2 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 200 μl of Calcium chloride (1 M) 150 μl of Polyethylene glycol 400 (100 v/v) 550 μl of water (100 v/v) |
C3 |
| pH 6.5 | 100 μl of 2-Propanol (100 v/v) 250 μl of Polyethylene glycol 400 (100 v/v) 100 μl of MES pH 6.5 (1 M) 550 μl of water (100 v/v) |
C4 |
| pH 8.5 | 250 μl of Polyethylene glycol 400 (100 v/v) 75 μl of tri-Sodium citrate (2 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 575 μl of water (100 v/v) |
C5 |
| pH 4.6 | 100 μl of Ethylene glycol (50 v/v) 100 μl of Sodium acetate pH 4.6 (1 M) 150 μl of Polyethylene glycol monomethyl ether 550 (100 v/v) 650 μl of water (100 v/v) |
C6 |
| pH 9 | 100 μl of BICINE pH 9 (1 M) 100 μl of Sodium chloride (1 M) 200 μl of Polyethylene glycol monomethyl ether 550 (100 v/v) 600 μl of water (100 v/v) |
C7 |
| pH 8.5 | 10 μl of Dithiothreitol (0.1 M) 400 μl of Polyethylene glycol 1,000 (50 w/v) 100 μl of tris chloride BCC pH 8.5 (1 M) 490 μl of water (100 v/v) |
C8 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 16 μl of Lithium sulfate (3 M) 700 μl of Polyethylene glycol 1,000 (50 w/v) 183 μl of water (100 v/v) |
C9 |
| pH 6.5 | 240 μl of Polyethylene glycol 2,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 100 μl of Magnesium acetate (2 M) 560 μl of water (100 v/v) |
C10 |
| pH 4.6 | 40 μl of Magnesium chloride (2.5 M) 100 μl of Sodium acetate pH 4.6 (1 M) 500 μl of Polyethylene glycol 2,000 (50 w/v) 360 μl of water (100 v/v) |
C11 |
| pH 4.6 | 20 μl of Magnesium chloride (2.5 M) 100 μl of Sodium acetate pH 4.6 (1 M) 600 μl of Polyethylene glycol 2,000 (50 w/v) 280 μl of water (100 v/v) |
C12 |
| pH 5 | 480 μl of Polyethylene glycol monomethyl ether 2,000 (50 w/v) 100 μl of Sodium phosphate citrate pH 5 (1 M) 420 μl of water (100 v/v) |
D1 |
| pH 6.5 | 240 μl of Polyethylene glycol 3,350 (50 w/v) 100 μl of Sodium chloride (5 M) 100 μl of MES pH 6.5 (1 M) 560 μl of water (100 v/v) |
D2 |
| pH 5.6 | 240 μl of Polyethylene glycol 3,350 (50 w/v) 50 μl of tri-Sodium citrate pH 5.6 (1 M) 66 μl of Ammonium sulfate (3 M) 50 μl of Magnesium sulfate (1 M) 593 μl of water (100 v/v) |
D3 |
| pH 7.5 | 10 μl of Cadmium chloride (1 M) 100 μl of Imidazole pH 7.5 (1 M) 300 μl of Polyethylene glycol 3,350 (50 w/v) 83 μl of Ammonium sulfate (3 M) 506 μl of water (100 v/v) |
D4 |
| pH 7 | 400 μl of Polyethylene glycol 3,350 (50 w/v) 150 μl of di-Sodium L-malate pH 7 (1 M) 450 μl of water (100 v/v) |
D5 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 400 μl of Polyethylene glycol 3,350 (50 w/v) 40 μl of Sodium chloride (5 M) 100 μl of L-Glutathione reduced (0.2 M) 360 μl of water (100 v/v) |
D6 |
| pH 8.5 | 400 μl of Polyethylene glycol 3,350 (50 w/v) 24 μl of Sodium chloride (5 M) 50 μl of Dithiothreitol (0.1 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 426 μl of water (100 v/v) |
D7 |
| NA | 400 μl of Polyethylene glycol 3,350 (50 w/v) 200 μl of Potassium nitrate (1 M) 400 μl of water (100 v/v) |
D8 |
| NA | 440 μl of Polyethylene glycol 3,350 (50 w/v) 40 μl of Ammonium formate (2.5 M) 520 μl of water (100 v/v) |
D9 |
| pH 5 | 480 μl of Polyethylene glycol 3,350 (50 w/v) 100 μl of tri-Sodium citrate pH 5 (1 M) 420 μl of water (100 v/v) |
D10 |
| pH 4.6 | 600 μl of Polyethylene glycol 3,350 (50 w/v) 100 μl of Sodium acetate pH 4.6 (1 M) 40 μl of Ammonium acetate (5 M) 260 μl of water (100 v/v) |
D11 |
| pH 5.6 | 200 μl of Ammonium acetate pH 5.6 (1 M) 200 μl of 2-Propanol (100 v/v) 40 μl of Calcium chloride (5 M) 375 μl of Polyethylene glycol 3,350 (80 w/v) 185 μl of water (100 v/v) |
D12 |
| pH 8.5 | 650 μl of Polyethylene glycol 3,350 (50 w/v) 80 μl of Magnesium chloride (2.5 M) 100 μl of Sodium chloride (5 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 70 μl of water (100 v/v) |
E1 |
| pH 6.5 | 160 μl of Polyethylene glycol 4,000 (50 w/v) 4 μl of Magnesium chloride (2.5 M) 50 μl of MES pH 6.5 (1 M) 100 μl of Dithiothreitol (0.1 M) 686 μl of water (100 v/v) |
E2 |
| pH 7 | 50 μl of PIPES pH 7 (1 M) 200 μl of Polyethylene glycol 4,000 (50 w/v) 100 μl of Dithiothreitol (0.1 M) 650 μl of water (100 v/v) |
E3 |
| pH 7.5 | 200 μl of Polyethylene glycol 4,000 (50 w/v) 100 μl of HEPES pH 7.5 (1 M) 150 μl of Ethylene glycol (100 v/v) 80 μl of Magnesium chloride (2.5 M) 100 μl of 2-Propanol (100 v/v) 370 μl of water (100 v/v) |
E4 |
| pH 7.5 | 200 μl of Polyethylene glycol 4,000 (50 w/v) 100 μl of HEPES pH 7.5 (1 M) 700 μl of water (100 v/v) |
E5 |
| pH 7.5 | 300 μl of Polyethylene glycol 4,000 (50 w/v) 100 μl of HEPES pH 7.5 (1 M) 100 μl of 2-Propanol (100 v/v) 500 μl of water (100 v/v) |
E6 |
| pH 8.5 | 300 μl of Polyethylene glycol 4,000 (50 w/v) 37 μl of Sodium acetate (2 M) 20 μl of Polyethylene glycol 6,000 (50 w/v) 200 μl of Sodium chloride (1 M) 75 μl of tris chloride BCC pH 8.5 (1 M) 367 μl of water (100 v/v) |
E7 |
| pH 5.5 | 300 μl of Polyethylene glycol 4,000 (50 w/v) 31 μl of di-Sodium DL-malate pH 7 (3 M) 200 μl of Ammonium sulfate (1 M) 1 μl of di-Sodium DL-malate pH 5 (3 M) 466 μl of water (100 v/v) |
E8 |
| pH 6.5 | 400 μl of Polyethylene glycol 4,000 (50 w/v) 100 μl of BIS-TRIS pH 6.5 (1 M) 100 μl of Sodium chloride (1 M) 400 μl of water (100 v/v) |
E9 |
| pH 7.5 | 400 μl of Polyethylene glycol 4,000 (50 w/v) 100 μl of HEPES pH 7.5 (1 M) 80 μl of Magnesium chloride (2.5 M) 420 μl of water (100 v/v) |
E10 |
| pH 8.5 | 400 μl of Polyethylene glycol 4,000 (50 w/v) 80 μl of Magnesium chloride (2.5 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 420 μl of water (100 v/v) |
E11 |
| pH 6.5 | 500 μl of Polyethylene glycol 4,000 (50 w/v) 80 μl of Magnesium chloride (2.5 M) 100 μl of MES pH 6.5 (1 M) 320 μl of water (100 v/v) |
E12 |
| pH 8.5 | 500 μl of Polyethylene glycol 4,000 (50 w/v) 33 μl of Lithium sulfate (3 M) 100 μl of tris chloride BCC pH 8.5 (1 M) 366 μl of water (100 v/v) |
F1 |
| pH 7.5 | 200 μl of Lithium acetate pH 7.5 (1 M) 560 μl of Polyethylene glycol 4,000 (50 w/v) 240 μl of water (100 v/v) |
F2 |
| pH 6.5 | 600 μl of Polyethylene glycol 4,000 (50 w/v) 100 μl of Sodium acetate (2 M) 100 μl of MES pH 6.5 (1 M) 200 μl of water (100 v/v) |
F3 |
| pH 8.5 | 600 μl of Polyethylene glycol 4,000 (50 w/v) 66 μl of Ammonium sulfate (3 M) 150 μl of tris chloride BCC pH 8.5 (1 M) 183 μl of water (100 v/v) |
F4 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 160 μl of Polyethylene glycol monomethyl ether 5,000 (50 w/v) 100 μl of 2-Propanol (100 v/v) 640 μl of water (100 v/v) |
F5 |
| pH 6.5 | 500 μl of Polyethylene glycol monomethyl ether 5,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 66 μl of Ammonium sulfate (3 M) 333 μl of water (100 v/v) |
F6 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 600 μl of Polyethylene glycol monomethyl ether 5,000 (50 w/v) 66 μl of Ammonium sulfate (3 M) 233 μl of water (100 v/v) |
F7 |
| pH 6.5 | 600 μl of Polyethylene glycol monomethyl ether 5,000 (50 w/v) 100 μl of ADA pH 6.5 (1 M) 33 μl of Ammonium sulfate (3 M) 266 μl of water (100 v/v) |
F8 |
| pH 6.5 | 400 μl of Polyethylene glycol 6,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 500 μl of water (100 v/v) |
F9 |
| pH 6.5 | 560 μl of Polyethylene glycol 6,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 100 μl of Dithiothreitol (0.1 M) 240 μl of water (100 v/v) |
F10 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 600 μl of Polyethylene glycol 6,000 (50 w/v) 58 μl of Lithium sulfate (3 M) 241 μl of water (100 v/v) |
F11 |
| pH 7 | 100 μl of PIPES pH 7 (1 M) 600 μl of Polyethylene glycol 6,000 (50 w/v) 100 μl of Dithiothreitol (0.1 M) 200 μl of water (100 v/v) |
F12 |
| pH 6.5 | 640 μl of Polyethylene glycol 6,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 260 μl of water (100 v/v) |
G1 |
| pH 6.5 | 200 μl of Ethylene glycol (100 v/v) 140 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 560 μl of water (100 v/v) |
G2 |
| pH 6.5 | 75 μl of Calcium acetate (2 M) 160 μl of Ethylene glycol (100 v/v) 140 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 525 μl of water (100 v/v) |
G3 |
| pH 8.5 | 100 μl of Polyethylene glycol 200 (100 v/v) 200 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of tris chloride BCC pH 8.5 (1 M) 600 μl of water (100 v/v) |
G4 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 240 μl of Polyethylene glycol 8,000 (50 w/v) 660 μl of water (100 v/v) |
G5 |
| pH 8.5 | 125 μl of di-Sodium tartrate (2 M) 240 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of tris chloride BCC pH 8.5 (1 M) 535 μl of water (100 v/v) |
G6 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 50 μl of Potassium di-hydrogen phosphate (2 M) 320 μl of Polyethylene glycol 8,000 (50 w/v) 530 μl of water (100 v/v) |
G7 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 40 μl of Ethylene glycol (50 v/v) 320 μl of Polyethylene glycol 6,000 (50 w/v) 30 μl of Sodium chloride (5 M) 510 μl of water (100 v/v) |
G8 |
| pH 6.5 | 360 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 100 μl of Magnesium acetate (2 M) 440 μl of water (100 v/v) |
G9 |
| pH 6.5 | 360 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 540 μl of water (100 v/v) |
G10 |
| pH 8.5 | 360 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of tris chloride BCC pH 8.5 (1 M) 540 μl of water (100 v/v) |
G11 |
| pH 5 | 100 μl of tri-Sodium citrate pH 5 (1 M) 400 μl of Polyethylene glycol 8,000 (50 w/v) 50 μl of Magnesium acetate (2 M) 450 μl of water (100 v/v) |
G12 |
| pH 8.5 | 20 μl of Ethylene glycol (100 v/v) 80 μl of Magnesium chloride (2.5 M) 400 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of tris chloride BCC pH 8.5 (1 M) 400 μl of water (100 v/v) |
H1 |
| pH 8.5 | 20 μl of Ethylene glycol (100 v/v) 440 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of tris chloride BCC pH 8.5 (1 M) 440 μl of water (100 v/v) |
H2 |
| pH 4.6 | 20 μl of Magnesium chloride (2.5 M) 100 μl of Sodium acetate pH 4.6 (1 M) 500 μl of Polyethylene glycol 8,000 (50 w/v) 380 μl of water (100 v/v) |
H3 |
| pH 6.5 | 80 μl of 1,3-Propanediol (50 v/v) 600 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 66 μl of Ammonium sulfate (3 M) 153 μl of water (100 v/v) |
H4 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 600 μl of Polyethylene glycol 8,000 (50 w/v) 200 μl of Glycerol (100 v/v) 100 μl of Dithiothreitol (0.1 M) |
H5 |
| pH 6.5 | 180 μl of Polyethylene glycol 8,000 (50 w/v) 100 μl of Zinc acetate (2 M) 100 μl of MES pH 6.5 (1 M) 620 μl of water (100 v/v) |
H6 |
| pH 6.5 | 100 μl of BIS-TRIS pH 6.5 (1 M) 320 μl of Polyethylene glycol 10,000 (50 w/v) 100 μl of Ethylene glycol (50 v/v) 100 μl of Ammonium sulfate (3 M) 380 μl of water (100 v/v) |
H7 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 200 μl of Polyethylene glycol 10,000 (50 w/v) 80 μl of Ethylene glycol (100 v/v) 620 μl of water (100 v/v) |
H8 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 300 μl of Polyethylene glycol 10,000 (50 w/v) 50 μl of Dithiothreitol (0.1 M) 550 μl of water (100 v/v) |
H9 |
| pH 8.5 | 300 μl of Polyethylene glycol 10,000 (50 w/v) 100 μl of tris chloride BCC pH 8.5 (1 M) 600 μl of water (100 v/v) |
H10 |
| pH 6.5 | 240 μl of Polyethylene glycol 20,000 (50 w/v) 100 μl of MES pH 6.5 (1 M) 660 μl of water (100 v/v) |
H11 |
| pH 7.5 | 100 μl of HEPES pH 7.5 (1 M) 200 μl of Polyethylene glycol 20,000 (50 w/v) 40 μl of Ammonium formate (2.5 M) 660 μl of water (100 v/v) |
H12 |
| NA | 100 μl of Potassium hydrogen tartrate (0.1 M) 300 μl of Polyethylene glycol 20,000 (50 w/v) 600 μl of water (100 v/v) |